Flupirtine maleate has a triple effect of analgesic, muscle relaxation and neuroprotective, and has an analgesic effect on pain caused by various causes.
Flupirtine maleate has triple effects of relieving pain, relaxing muscles and protecting nerves. Its mechanism of action: (1) selectively activates voltage-gated potassium channels on nerve cell membranes, promotes potassium outflow, stabilizes cell membrane potential, indirectly inhibits NMDA receptors, blocks NMDA receptor-mediated calcium influx, buffers the sensitive effect of increased calcium ion concentration in cells, and blocks the conduction of pain impulses. (2) Enhance the long-term inhibition of synaptic transmission, block the conduction of nerve signals, and interrupt the connection bond of chronic pain center sensitization. (3) Inhibit the input of stimulation signals of the spine, subcortical layer and cortical layer, and activate the norepinephric neurosuppressive system of the spine and subcortical layer.
|Appearance||White powder||White powder|
|Package details:||1kg/foil bag,25kg/drum|
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